Scientific Reports, 9(1), 20056 (2019)
Hirakawa, Tomoko; Nasu, Kaei; Miyabe, Saori; Kouji, Hiroyuki; Katoh, Akira; Uemura, Naoto; Narahara, Hisashi
アーカイブ: ニュース
mS-11, a mimetic of the mSin3-binding helix in NRSF, ameliorates social interaction deficits in a prenatal valproic acid-induced autism mouse model
Pharmacology Biochemistry and Behavior, 176, 1-5 (2019)
Kawase, Haruki; Ago, Yukio; Naito, Megumi; Higuchi, Momoko; Hara, Yuta; Hasebe, Shigeru; Tsukada, Shinji; Kasai, Atsushi; Nakazawa, Takanobu; Mishina, Tadashi; Kouji, Hiroyuki; Takuma, Kazuhiro; Hashimoto, Hitoshi
The novel inhibitor PRI-724 for Wnt/β-catenin/CBP signaling ameliorates bleomycin-induced pulmonary fibrosis in mice
Experimental Lung Research, 45(7), 188-199 (2019)
Okazaki, Hiroyasu; Sato, Seidai; Koyama, Kazuya; Morizumi, Shun; Abe, Shuichi; Azuma, Momoyo; Chen, Yajuan; Goto, Hisatsugu; Aono, Yoshinori; Ogawa, Hirohisa; Kagawa, Kozo; Nishimura, Haruka; Kawano, Hiroshi; Toyoda, Yuko; Uehara, Hisanori; Kouji, Hiroyuki; Nishioka, Yasuhiko
A mimetic of the mSin3-binding helix of NRSF/REST ameliorates abnormal pain behavior in chronic pain models
Bioorganic and Medicinal Chemistry Letters, 27, 4705-4709 (2017)
Ueda, Hiroshi; Jun-ichi Kurita; Neyama, Hiroyuki; Hirao, Yuuka; Kouji, Hiroyuki; Mishina, Tadashi; Kasai, Masaji; Nakano, Hirofumi; Yoshimori, Atsushi; Nishimura, Yoshifumi
Establishment of an intermittent cold stress model using Tupaia Belangeri and evaluation of compound C737 targeting neuron-restrictive silencer factor
Experimental Animals, 65(3), 285-292 (2016)
Hai-Ying, Chi; Nagano, Kiori; Ezzikouri, Sayeh; Yamaguchi, Chiho; Kayesh, Mohammad Enamul Hoque; Rebbani, Khadija; Kitab, Bouchra; Nakano, Hirohumi; Kouji, Hiroyuki; Kohara, Michinori; Tsukiyama-Kohara, Kyoko
Follow-up: Prospective compound design using the ‘SAR Matrix’ method and matrix-derived conditional probabilities of activity
F1000Research, 4, 75 (2015)
Gupta-Ostermann, Disha; Hirose, Yoichiro; Odagami, Takenao; Kouji, Hiroyuki; Bajorath, Jurgen
Three-dimensional structural diversity-oriented peptidomimetics based on the cyclopropylic strain
Organic Letters, 15(7), 1686-1689 (2013)
Mizuno, Akira; Miura, Shiho; Watanabe, Mizuki; Ito, Yoshihiko; Yamada, Shizuo; Odagami, Takenao; Kogami, Yuji; Arisawa, Mitsuhiro; Shuto, Satoshi
Protein-Protein Interaction をターゲットとした創薬
Medchem News, 22(1), 21-24 (2012) (Japanese)
Odagami, Takenao; Kouji, Hiroyuki
Deprotection of Nin-formyl group on tryptophan by application of new reagent, 1,2-dimethylethylendiamine in aqueous solution
Advances in Experimental Medicine and Biology, 611, 159-160 (2009)
Odagami, Takenao; Kogami, Yuji; Kouji, Hiroyuki; Tsuda, Yuko; Okada, Yoshio
Identification of new agonists of urotensin-II from a cyclic peptide library
Bioorganic and Medicinal Chemistry, 17, 6742-6747 (2009)
Odagami, Takenao; Tsuda, Yuko; Kogami, Yuji; Kouji, Hiroyuki; Okada, Yoshio